Found 890 of ic50 for ALPHA-1D ADRENERGIC RECEPTOR
having polymerids = 7476,7889,49000208 and
complexids = 50002812,50000229,50000717,50006003
having polymerids = 7476,7889,49000208 and
complexids = 50002812,50000229,50000717,50006003
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 0.00692nMAssay Description:Binding affinity at Alpha-1 adrenergic receptor sites on rat cerebral cortical membranes by [3H]prazosin displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Antagonist activity at alpha-1D adrenergic receptor (unknown origin) transfected in HEK293 cells assessed as reduction in agonist-induced calcium mob...More data for this Ligand-Target Pair
Affinity DataIC50: 0.150nMAssay Description:Antagonist activity at human alpha1D receptor transfected in HEK293 cells co-transfected with Galpha16 assessed as reduction in intracellular calcium...More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 0.162nMAssay Description:Displacement of [3H]prazosin binding to Alpha-1 adrenergic receptor sites on rat cerebral cortical membranes at 100 nM concentrationMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 0.180nMAssay Description:Ability to inhibit binding of [3H]PRAZ to alpha-1 adrenergic receptor in rat brainMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 0.25nMAssay Description:Displacement of [3H]-prazosin from rat alpha1 adrenoceptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity at alpha-1D adrenergic receptor (unknown origin) transfected in HEK293 cells assessed as reduction in agonist-induced calcium mob...More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 0.360nMAssay Description:Inhibition of [3H]prazosin binding to alpha-1 adrenergic receptor from rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at alpha-1D adrenergic receptor (unknown origin) transfected in HEK293 cells assessed as reduction in agonist-induced calcium mob...More data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at alpha-1D adrenergic receptor (unknown origin) transfected in HEK293 cells assessed as reduction in agonist-induced calcium mob...More data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at alpha-1D adrenergic receptor (unknown origin) transfected in HEK293 cells assessed as reduction in agonist-induced calcium mob...More data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at alpha-1D adrenergic receptor (unknown origin) transfected in HEK293 cells assessed as reduction in agonist-induced calcium mob...More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 0.450nMAssay Description:Ability to inhibit binding of [3H]PRAZ to alpha-1 adrenergic receptor in rat brainMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 0.513nMAssay Description:Binding affinity at Alpha-1 adrenergic receptor sites on rat cerebral cortical membranes by [3H]prazosin displacement.More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 0.580nMAssay Description:Inhibition of specific [3H]prazosin binding (0.2 nM) to rat brain membranes alpha1 adrenoceptor.More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Alpha-1-adrenolytic activity was assessed from the ability to inhibit [3H]prazosin binding to rat cerebral cortex preparationMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 0.690nMAssay Description:Ability to bind at alpha-1 adrenergic receptor by displacing [3H]WB-4101More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 0.692nMAssay Description:Displacement of [3H]prazosin binding to Alpha-1 adrenergic receptor sites on rat cerebral cortical membranes at 100 nM concentrationMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 0.876nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in rat cerebral cortex tissue using [3H]WB-4101 as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:In vitro affinity for cortical alpha-1 adrenergic receptor labelled with [3H]WB-4101More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:In vitro affinity for cortical alpha-1 adrenergic receptor labelled with [3H]WB-4101More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Ability to bind at alpha-1 adrenergic receptor by displacing [3H]WB-4101More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Ability to bind at alpha-1 adrenergic receptor by displacing [3H]WB-4101More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Homo sapiens (Human))
Panjab University
Curated by ChEMBL
Panjab University
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity at Adrenergic alpha-1 receptor (unknown origin)More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Homo sapiens (Human))
Panjab University
Curated by ChEMBL
Panjab University
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity at Adrenergic alpha-1 receptor (unknown origin)More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in rat cerebral cortex tissue using [3H]WB-4101 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Antagonist activity at human full-length N-terminal SNAP-tagged alpha1D adrenoceptor expressed in HEK293 cells assessed as inhibition of agonist-indu...More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Ability to inhibit binding of [3H]PRAZ to alpha-1 adrenergic receptor in rat brainMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Compound is evaluated for its ability to compete with [3H]prazosin for binding to Alpha-1 adrenergic receptor sites on rat cerebral cortical membrane...More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in rat cerebral cortex tissue using [3H]WB-4101 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Antagonist activity at alpha-1D adrenergic receptor (unknown origin) transfected in HEK293 cells assessed as reduction in agonist-induced calcium mob...More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mus musculus (Mouse))
The Australian Nuclear Science And Technology Organisation
Curated by ChEMBL
The Australian Nuclear Science And Technology Organisation
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenoceptor in C57BL/6 mouse hippocampal homogenates after 40 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:In vitro affinity for cortical alpha-1 adrenergic receptor labelled with [3H]WB-4101More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:In vitro affinity for cortical alpha-1 adrenergic receptor labelled with [3H]WB-4101More data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Displacement of [3H]-Prazosin from human alpha-1D adrenergic receptor transfected in CHO cell membranes after 2 hrs by microplate scintillation count...More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of whole rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 2.5nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in rat cerebral cortex tissue using [3H]WB-4101 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Antagonist activity at alpha-1D adrenergic receptor (unknown origin) transfected in HEK293 cells assessed as reduction in agonist-induced calcium mob...More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 2.60nMAssay Description:Displacement of [3H]prazosin from alpha-1 adrenoceptors in whole rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:In vitro affinity for cortical alpha-1 adrenergic receptor labelled with [3H]WB-4101More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of whole rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1D-adrenoreceptors on isolated thoracic aorta from ratMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 3.40nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of whole rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 3.40nMAssay Description:Binding affinity at Alpha-1 adrenergic receptor sites on rat cerebral cortical membranes by [3H]prazosin displacement.More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 3.40nMAssay Description:Displacement of [3H]prazosin binding to Alpha-1 adrenergic receptor sites on rat cerebral cortical membranes at 100 nM concentrationMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:In vitro affinity for cortical alpha-1 adrenergic receptor labelled with [3H]WB-4101More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 4.40nMAssay Description:Displacement of [3H]prazosin binding to Alpha-1 adrenergic receptor sites on rat cerebral cortical membranes at 100 nM concentrationMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
National Institute On Aging/Grc
Curated by ChEMBL
National Institute On Aging/Grc
Curated by ChEMBL
Affinity DataIC50: 4.5nMAssay Description:Displacement of [3H]prazosin binding to Alpha-1 adrenergic receptor sites on rat cerebral cortical membranes at 100 nM concentrationMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Antagonist affinity [non competitive (irreversible)] at alpha-1D-adrenoreceptors on isolated thoracic aorta from ratMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Homo sapiens (Human))
Panjab University
Curated by ChEMBL
Panjab University
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Antagonist activity at Adrenergic alpha-1 receptor in human Prostate cell in presence of (125I)-Heat by Competitive binding assayMore data for this Ligand-Target Pair